JH-XI-10-02, CAS [[2209085-22-1]]

Artikelnummer: MCE-HY-111518
Artikelname: JH-XI-10-02, CAS [[2209085-22-1]]
Artikelnummer: MCE-HY-111518
Hersteller Artikelnummer: HY-111518
Alternativnummer: MCE-HY-111518-5MG,MCE-HY-111518-10MG,MCE-HY-111518-1MG,MCE-HY-111518-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
JH-XI-10-02 is a PROTAC connected by ligands for Cereblon and CDK. JH-XI-10-02 is a highly potent and selective PROTAC CDK8 degrader, with an IC50 of 159 nM. JH-XI-10-02 causes proteasomal degradation, does not affect CDK8 mRNA levels. JH-XI-10-02 shows no effect on CDK19[1].
Molekulargewicht: 920.14
Reinheit: 99.73
CAS Nummer: [2209085-22-1]
Formel: C53H69N5O9
Target-Kategorie: CDK,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound