M3258, CAS [[2285330-15-4]]

Produktübersicht

• Artikelname: M3258, CAS [[2285330-15-4]]
• Artikelnummer: MCE-HY-111790
• Hersteller Artikelnummer: HY-111790
• Alternativnummer: MCE-HY-111790-10MMX1ML,MCE-HY-111790-10MG,MCE-HY-111790-100MG,MCE-HY-111790-5MG,MCE-HY-111790-50MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

M3258 is an orally bioavailable, potent, reversible and highly selective immunoproteasome subunit LMP7 (beta5i) inhibitor. M3258 exerts high biochemical (IC50=3.6 nM) and cellular (IC50=3.4 nM) potency against the LMP7 subunit. M3258 shows strong antitumor efficacy in multiple myeloma xenograft models. M3258 leads to a significant and prolonged suppression of tumor LMP7 activity and ubiquitinated protein turnover and the induction of apoptosis in multiple myeloma cells[1][2].

Produkteigenschaften

• Molekulargewicht: 329.16
• Reinheit: 98
• CAS Nummer: [2285330-15-4]
• Formel: C17H20BNO5
• Target-Kategorie: Apoptosis,Proteasome

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound