CB1 antagonist 4, CAS [[1253641-65-4]]

Artikelnummer: MCE-HY-112340
Artikelname: CB1 antagonist 4, CAS [[1253641-65-4]]
Artikelnummer: MCE-HY-112340
Hersteller Artikelnummer: HY-112340
Alternativnummer: MCE-HY-112340-100MG,MCE-HY-112340-10MMX1ML,MCE-HY-112340-5MG,MCE-HY-112340-10MG,MCE-HY-112340-50MG,MCE-HY-112340-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
CB1 antagonist 4 (compound 8) is a selective cannabinoid receptor 1 (CB1) inverse agonist with an IC50 of 8.5 nM for human CB1. CB1 antagonist 4 shows selective for CB1 over CB2 receptors (IC50 of 604.9 nM). CB1 antagonist 4 inhibits GTP binding to CB1-overexpressing cell membranes with an EC50 of 18.5 nM[1].
Molekulargewicht: 617.51
Reinheit: 98.00
CAS Nummer: [1253641-65-4]
Formel: C30H25Cl2F3N4OS
Target-Kategorie: Cannabinoid Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound