PROTAC TBK1 degrader-2, CAS [[2052306-13-3]]

Artikelnummer: MCE-HY-112557
Artikelname: PROTAC TBK1 degrader-2, CAS [[2052306-13-3]]
Artikelnummer: MCE-HY-112557
Hersteller Artikelnummer: HY-112557
Alternativnummer: MCE-HY-112557-1MG,MCE-HY-112557-5MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC TBK1 degrader-2 is a Ligands for Target Protein for PROTAC. PROTAC TBK1 degrader-2 is a potent degrader based on the serine/threonine kinase TANK-binding kinase 1 (TBK1) (DC50=15 nM, Kd=4.6 nM) with a maximum efficiency of 96%. PROTAC TBK1 degrader-2 also targets to IkB kinase IKKepsilon (IC50=8.7 nM), with low selectivity over TBK1 (IC50=1.3 nM)[1].
Molekulargewicht: 1093.18
Reinheit: 98.20
CAS Nummer: [2052306-13-3]
Formel: C53H74BrN9O9S
Target-Kategorie: IKK,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound