PROTAC TBK1 degrader-2 is a Ligands for Target Protein for PROTAC. PROTAC TBK1 degrader-2 is a potent degrader based on the serine/threonine kinase TANK-binding kinase 1 (TBK1) (DC50=15 nM, Kd=4.6 nM) with a maximum efficiency of 96%. PROTAC TBK1 degrader-2 also targets to IkB kinase IKKepsilon (IC50=8.7 nM), with low selectivity over TBK1 (IC50=1.3 nM)[1].
Molecular Weight:
1093.18
Purity:
98.20
CAS Number:
[2052306-13-3]
Formula:
C53H74BrN9O9S
Target:
IKK,PROTACs
Application Notes:
MCE Product type: Reference compound
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