GSK8814, CAS [[1997369-78-4]]

Produktübersicht

• Artikelname: GSK8814, CAS [[1997369-78-4]]
• Artikelnummer: MCE-HY-114204
• Hersteller Artikelnummer: HY-114204
• Alternativnummer: MCE-HY-114204-5MG,MCE-HY-114204-10MG,MCE-HY-114204-1MG,MCE-HY-114204-10MMX1ML
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

GSK8814 is a potent and selective ATAD2 bromodomain chemical probe and inhibitor (IC50 = 0.059 µM), with a binding constant pKd = 8.1 and a pKi = 8.9 in BROMOscan. GSK8814 binds to ATAD2 and BRD4 BD1 with pIC50s of 7.3 and 4.6, respectively. GSK8814 shows 500-fold selectivity for ATAD2 over BRD4 BD1. GSK8814 can be researched for cancer associated with ATAD2 bromodomain[1][2][3].

Produkteigenschaften

• Molekulargewicht: 527.61
• Reinheit: 99.80
• CAS Nummer: [1997369-78-4]
• Formel: C28H35F2N5O3
• Target-Kategorie: Epigenetic Reader Domain

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound