VU041, CAS [[332943-64-3]]

Artikelnummer: MCE-HY-118607
Artikelname: VU041, CAS [[332943-64-3]]
Artikelnummer: MCE-HY-118607
Hersteller Artikelnummer: HY-118607
Alternativnummer: MCE-HY-118607-5MG,MCE-HY-118607-10MMX1ML,MCE-HY-118607-50MG,MCE-HY-118607-10MG,MCE-HY-118607-25MG,MCE-HY-118607-100MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
VU041 is a first submicromolar-affinity inhibitor of Anopheles (An.) gambiae and Aedes (Ae.) aegypti inward rectifier potassium 1 (Kir1) channels with IC50 values of 2.5 µM and 1.7 µM, respectively. VU041 inhibits appreciably is mammalian Kir2.1 (IC50 of 12.7 µM), and has less inhibitory effect on mammalian Kir1.1, Kir4.1, Kir6.2/SUR1, and Kir7.1. VU041 also induces impaired Malpighian tubule function[1].
Molekulargewicht: 363.38
Reinheit: 99.31
CAS Nummer: [332943-64-3]
Formel: C19H20F3N3O
Target-Kategorie: Parasite,Potassium Channel
Anwendungsbeschreibung: MCE Product type: Reference compound