Genz-669178, CAS [[1254834-91-7]] Preis auf Anfrage

Artikelnummer: MCE-HY-120462
Artikelname: Genz-669178, CAS [[1254834-91-7]] Preis auf Anfrage
Artikelnummer: MCE-HY-120462
Hersteller Artikelnummer: HY-120462
Alternativnummer: MCE-HY-120462-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Genz-669178 is an inhibitor for dihydroorotate dehydrogenase (DHODH) with IC50 of 0.015-0.05 µM in Plasmodium spp.. Genz-669178 inhibits P. berghei, P. falciparum strains 3D7 and Dd2 with IC50 of 0.068, 0.008 and 0.01 µM, respectively. Genz-669178 exhibits anti-malarial efficacy in P. berghei-infected mice with ED50 of 13-21 mg/kg/day. Genz-669178 exhibits good pharmacokinetic characteristics in mice[1].
Molekulargewicht: 322.38
CAS Nummer: [1254834-91-7]
Formel: C17H14N4OS
Target-Kategorie: Dihydroorotate Dehydrogenase,Parasite
Anwendungsbeschreibung: MCE Product type: Reference compound