hSMG-1 inhibitor 11j, CAS [[1402452-15-6]]

Artikelnummer: MCE-HY-124719
Artikelname: hSMG-1 inhibitor 11j, CAS [[1402452-15-6]]
Artikelnummer: MCE-HY-124719
Hersteller Artikelnummer: HY-124719
Alternativnummer: MCE-HY-124719-5MG,MCE-HY-124719-10MMX1ML,MCE-HY-124719-25MG,MCE-HY-124719-50MG,MCE-HY-124719-100MG,MCE-HY-124719-1MG,MCE-HY-124719-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
hSMG-1 inhibitor 11j, a pyrimidine derivative, is a potent and selective inhibitor of hSMG-1, with an IC50 of 0.11 nM. hSMG-1 inhibitor 11j exhibits >455-fold selectivity for hSMG-1 over mTOR (IC50=50 nM), PI3Kalpha/gamma (IC50=92/60 nM) and CDK1/CDK2 (IC50=32/7.1 µM). hSMG-1 inhibitor 11j can be used for the research of cancer[1].
Molekulargewicht: 566.07
Reinheit: 99.82
CAS Nummer: [1402452-15-6]
Formel: C27H28ClN7O3S
Target-Kategorie: CDK,GSK-3,mTOR,PI3K
Anwendungsbeschreibung: MCE Product type: Reference compound