Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (sigma1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 µM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain[1].
Molekulargewicht:
363.86
Reinheit:
99.47
CAS Nummer:
[1639220-17-9]
Formel:
C19H23ClFN3O
Target-Kategorie:
Potassium Channel,Sigma Receptor
Anwendungsbeschreibung:
MCE Product type: Reference compound1
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
