Sigma-1 receptor antagonist 3 (compound135) is a potent and selective Sigma-1 (sigma1) receptor antagonist with a Ki of 1.14 nM. Sigma-1 receptor antagonist 3 inhibits Human Ether-a-go-go-Related Gene (hERG) with an IC50 of 1.54 µM. Sigma-1 receptor antagonist 3 has the potential for the neuropathic pain[1].
Molecular Weight:
363.86
Purity:
99.47
CAS Number:
[1639220-17-9]
Formula:
C19H23ClFN3O
Target:
Potassium Channel,Sigma Receptor
Application Notes:
MCE Product type: Reference compound1
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