FGTI-2734, CAS [[1247018-19-4]]

Artikelnummer: MCE-HY-128350
Artikelname: FGTI-2734, CAS [[1247018-19-4]]
Artikelnummer: MCE-HY-128350
Hersteller Artikelnummer: HY-128350
Alternativnummer: MCE-HY-128350-25MG,MCE-HY-128350-5MG,MCE-HY-128350-10MG,MCE-HY-128350-10MMX1ML,MCE-HY-128350-50MG,MCE-HY-128350-100MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
FGTI-2734 is a RAS C-terminal mimetic dual farnesyl transferase (FT) and geranylgeranyl transferase-1 (GGT-1) inhibitor with IC50s of 250 nM and 520 nM for FT and GGT-1, respectively. FGTI-2734 can prevent membrane localization of KRAS, hence solving KRAS resistance problem and thwarting mutant KRAS patient-derived pancreatic tumors[1].
Molekulargewicht: 510.63
Reinheit: 99.85
CAS Nummer: [1247018-19-4]
Formel: C26H31FN6O2S
Target-Kategorie: Farnesyl Transferase
Anwendungsbeschreibung: MCE Product type: Reference compound