MRGPRX1 agonist 1, CAS [[2377379-39-8]]

Artikelnummer: MCE-HY-130118
Artikelname: MRGPRX1 agonist 1, CAS [[2377379-39-8]]
Artikelnummer: MCE-HY-130118
Hersteller Artikelnummer: HY-130118
Alternativnummer: MCE-HY-130118-5MG,MCE-HY-130118-25MG,MCE-HY-130118-10MG,MCE-HY-130118-50MG,MCE-HY-130118-100MG,MCE-HY-130118-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
MRGPRX1 agonist 1 is a highly potent MRGPRX1 agonist (EC50=50 nM) with greater than 50-fold selectivity for delta, µ, and kappa opioid receptors. MRGPRX1 agonist 1 is inactive against MRGPRC11. MRGPRC11 inhibits high voltage-activated (HVA) Ca2+ currents, reduces neurotransmitter release, and mitigates nociceptive transmission in the spinal cord. MRGPRX1 agonist 1 is useful for the study of chronic pain, especially neuropathic pain[1].
Molekulargewicht: 435.50
Reinheit: 99.95
CAS Nummer: [2377379-39-8]
Formel: C23H21N3O4S
Target-Kategorie: Mas-related G-protein-coupled Receptor (MRGPR)
Anwendungsbeschreibung: MCE Product type: Reference compound