MRGPRX1 agonist 1, CAS [[2377379-39-8]]

Product Overview

• Article Name: MRGPRX1 agonist 1, CAS [[2377379-39-8]]
• Biozol Catalog Number: MCE-HY-130118
• Supplier Catalog Number: HY-130118
• Alternative Catalog Number: MCE-HY-130118-5MG,MCE-HY-130118-25MG,MCE-HY-130118-10MG,MCE-HY-130118-50MG,MCE-HY-130118-100MG,MCE-HY-130118-10MMX1ML
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

MRGPRX1 agonist 1 is a highly potent MRGPRX1 agonist (EC50=50 nM) with greater than 50-fold selectivity for delta, µ, and kappa opioid receptors. MRGPRX1 agonist 1 is inactive against MRGPRC11. MRGPRC11 inhibits high voltage-activated (HVA) Ca2+ currents, reduces neurotransmitter release, and mitigates nociceptive transmission in the spinal cord. MRGPRX1 agonist 1 is useful for the study of chronic pain, especially neuropathic pain[1].

Product Properties

• Molecular Weight: 435.50
• Purity: 99.95
• CAS Number: [2377379-39-8]
• Formula: C23H21N3O4S
• Target: Mas-related G-protein-coupled Receptor (MRGPR)

Application Notes

• Application Notes: MCE Product type: Reference compound