PROTAC BRD2/BRD4 degrader-1, CAS [[2570470-42-5]] Preis auf Anfrage
Artikelnummer:
MCE-HY-130612
Hersteller Artikelnummer:
HY-130612
Alternativnummer:
MCE-HY-130612-1UNIT
Hersteller:
MedchemExpress
Kategorie:
Biochemikalien
PROTAC BRD2/BRD4 degrader-1 (compound 15) is a potent and selective BET protein BRD4 and BRD2 degrader, connected by ligands for Cereblon and BET. PROTAC BRD2/BRD4 degrader-1 rapidly induces reversible, long-lasting, and unexpectedly selective removal of BRD4 and BRD2 over BRD3. It effectively inhibits solid tumors with low cytotoxic effect. PROTAC BRD2/BRD4 degrader-1 is composed of the BET inhibitor, a linker, and the ligand thalidomide for cereblon (CRBN)/cullin 4A[1].
Molekulargewicht:
766.82
CAS Nummer:
[2570470-42-5]
Formel:
C39H38N6O9S
Target-Kategorie:
Epigenetic Reader Domain,PROTACs
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
