PROTAC BRD2/BRD4 degrader-1, CAS [[2570470-42-5]] Preis auf Anfrage

Catalog Number: MCE-HY-130612
Article Name: PROTAC BRD2/BRD4 degrader-1, CAS [[2570470-42-5]] Preis auf Anfrage
Biozol Catalog Number: MCE-HY-130612
Supplier Catalog Number: HY-130612
Alternative Catalog Number: MCE-HY-130612-1UNIT
Manufacturer: MedchemExpress
Category: Biochemikalien
PROTAC BRD2/BRD4 degrader-1 (compound 15) is a potent and selective BET protein BRD4 and BRD2 degrader, connected by ligands for Cereblon and BET. PROTAC BRD2/BRD4 degrader-1 rapidly induces reversible, long-lasting, and unexpectedly selective removal of BRD4 and BRD2 over BRD3. It effectively inhibits solid tumors with low cytotoxic effect. PROTAC BRD2/BRD4 degrader-1 is composed of the BET inhibitor, a linker, and the ligand thalidomide for cereblon (CRBN)/cullin 4A[1].
Molecular Weight: 766.82
CAS Number: [2570470-42-5]
Formula: C39H38N6O9S
Target: Epigenetic Reader Domain,PROTACs
Application Notes: MCE Product type: Reference compound1