K-Ras ligand-Linker Conjugate 4, CAS [[2378261-83-5]]

Artikelnummer: MCE-HY-130822
Artikelname: K-Ras ligand-Linker Conjugate 4, CAS [[2378261-83-5]]
Artikelnummer: MCE-HY-130822
Hersteller Artikelnummer: HY-130822
Alternativnummer: MCE-HY-130822-100MG,MCE-HY-130822-10MG,MCE-HY-130822-5MG,MCE-HY-130822-50MG,MCE-HY-130822-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
K-Ras ligand-Linker Conjugate 4 incorporates a ligand for K-Ras recruiting moiety, and a PROTAC linker, which recruit E3 ligases (such as VHL, CRBN, MDM2, and IAP). K-Ras ligand-Linker Conjugate 4 can be used in the synthesis of PROTAC K-Ras Degrader-1 (HY-129523), which is potent PROTAC K-Ras degrader that exhibits 70% degradation efficacy in SW1573 cells[1].
Molekulargewicht: 697.82
Reinheit: 98.76
CAS Nummer: [2378261-83-5]
Formel: C35H51N7O8
Target-Kategorie: Target Protein Ligand-Linker Conjugates
Anwendungsbeschreibung: MCE Product type: Reference compound