Androgen receptor antagonist 1, CAS [[1338812-36-4]]

Artikelnummer: MCE-HY-130992
Artikelname: Androgen receptor antagonist 1, CAS [[1338812-36-4]]
Artikelnummer: MCE-HY-130992
Hersteller Artikelnummer: HY-130992
Alternativnummer: MCE-HY-130992-25MG,MCE-HY-130992-5MG,MCE-HY-130992-50MG,MCE-HY-130992-10MG,MCE-HY-130992-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Androgen receptor antagonist 1 is an orally available full androgen receptor (AR) antagonist with an IC50 of 59 nM[1]. Androgen receptor antagonist 1 (Compound 6) can be used in the synthesis of PROTAC AR degraders, which results 24% and 47 % AR protein degradation in LNCaP cells at 1 µM and 10 µM, respectively[2].
Molekulargewicht: 416.90
Reinheit: 99.64
CAS Nummer: [1338812-36-4]
Formel: C21H25ClN4O3
Target-Kategorie: Androgen Receptor,Ligands for Target Protein for PROTAC
Anwendungsbeschreibung: Reference compound