M8891, CAS [[1464842-09-8]]

Artikelnummer: MCE-HY-133016
Artikelname: M8891, CAS [[1464842-09-8]]
Artikelnummer: MCE-HY-133016
Hersteller Artikelnummer: HY-133016
Alternativnummer: MCE-HY-133016-5MG,MCE-HY-133016-10MG,MCE-HY-133016-50MG,MCE-HY-133016-25MG,MCE-HY-133016-100MG,MCE-HY-133016-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
M8891 is an orally active, reversible and brain penetrant Methionine Aminopeptidase-2 (MetAP-2) inhibitor with an IC50 of 54 nM and a Ki of 4.33 nM. M8891 does not inhibit MetAP-1 (IC50>10 µM)[1]. M8891 inhibits growth of primary endothelial cells as well as tumor cells and demonstrates antiangiogenic and antitumoral activity[2].
Molekulargewicht: 385.36
Reinheit: 99.69
CAS Nummer: [1464842-09-8]
Formel: C20H17F2N3O3
Target-Kategorie: MetAP
Anwendungsbeschreibung: Reference compound