MS1943, CAS [[2225938-17-8]]

Produktübersicht

• Artikelname: MS1943, CAS [[2225938-17-8]]
• Artikelnummer: MCE-HY-133129
• Hersteller Artikelnummer: HY-133129
• Alternativnummer: MCE-HY-133129-100MG,MCE-HY-133129-25MG,MCE-HY-133129-500MG,MCE-HY-133129-1G,MCE-HY-133129-5MG,MCE-HY-133129-250MG,MCE-HY-133129-50MG,MCE-HY-133129-10MMX1ML,MCE-HY-133129-10MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

MS1943 is an orally active, PROTAC-based, selective degrader of EZH2 that effectively reduces EZH2 levels in cells. MS1943 has anticancer activity and exhibits cytotoxic effects in a variety of TNBC cells while sparing normal cells. In addition, MS1943 maintains high potency (IC50=120 nM) in inhibiting EZH2 methyltransferase activity and is highly selective for EZH2. (Structure Note: RED, EZH2 ligand (HY-148458), Blue, Hyt (HY-W001578))[1].

Produkteigenschaften

• Molekulargewicht: 718.93
• Reinheit: 98.92
• CAS Nummer: [2225938-17-8]
• Formel: C42H54N8O3
• Target-Kategorie: Apoptosis,Histone Methyltransferase,PROTACs

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound