Methocinnamox, CAS [[117339-76-1]] Preis auf Anfrage

Produktübersicht

• Artikelname: Methocinnamox, CAS [[117339-76-1]] Preis auf Anfrage
• Artikelnummer: MCE-HY-135698
• Hersteller Artikelnummer: HY-135698
• Alternativnummer: MCE-HY-135698-1UNIT
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: M-CAM

Produktbeschreibung

Methocinnamox (M-CAM) a selective and long-acting µ-opioid receptor (MOR) antagonist with a Ki of 0.6 nM. Methocinnamox binds to the orthosteric site of the MOR in a pseudo-irreversible, non-covalent manner, resulting in prolonged receptor blockade that persists until new receptors are synthesized. Methocinnamox acts as a reversible antagonist at both the kappa-opioid receptor (KOR) (Ki = 4.9 nM) and delta-opioid receptor (DOR) (Ki = 2.2 nM), and it exhibits no intrinsic agonist activity at these receptors. Methocinnamox can be used to reverse and prevent opioid overdose and addiction[1][2][3].

Produkteigenschaften

• Molekulargewicht: 484.59
• CAS Nummer: [117339-76-1]
• Formel: C30H32N2O4
• Target-Kategorie: Opioid Receptor

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound1