Methocinnamox, CAS [[117339-76-1]] Preis auf Anfrage

Product Overview

• Article Name: Methocinnamox, CAS [[117339-76-1]] Preis auf Anfrage
• Biozol Catalog Number: MCE-HY-135698
• Supplier Catalog Number: HY-135698
• Alternative Catalog Number: MCE-HY-135698-1UNIT
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: M-CAM

Product Description

Methocinnamox (M-CAM) a selective and long-acting µ-opioid receptor (MOR) antagonist with a Ki of 0.6 nM. Methocinnamox binds to the orthosteric site of the MOR in a pseudo-irreversible, non-covalent manner, resulting in prolonged receptor blockade that persists until new receptors are synthesized. Methocinnamox acts as a reversible antagonist at both the kappa-opioid receptor (KOR) (Ki = 4.9 nM) and delta-opioid receptor (DOR) (Ki = 2.2 nM), and it exhibits no intrinsic agonist activity at these receptors. Methocinnamox can be used to reverse and prevent opioid overdose and addiction[1][2][3].

Product Properties

• Molecular Weight: 484.59
• CAS Number: [117339-76-1]
• Formula: C30H32N2O4
• Target: Opioid Receptor

Application Notes

• Application Notes: MCE Product type: Reference compound1