BSJ-03-204 (triTFA)

Produktübersicht

• Artikelname: BSJ-03-204 (triTFA)
• Artikelnummer: MCE-HY-136250A
• Hersteller Artikelnummer: HY-136250A
• Alternativnummer: MCE-HY-136250A-10MG,MCE-HY-136250A-25MG,MCE-HY-136250A-5MG,MCE-HY-136250A-100MG,MCE-HY-136250A-50MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

BSJ-03-204 triTFA is a PROTAC connected by ligands for Cereblon and CDK. BSJ-03-204 triTFA is a potent and selective Palbociclib-based CDK4/6 dual degrader (PROTAC), with IC50s of 26.9 nM and 10.4 nM for CDK4/D1 and CDK6/D1, respectively. BSJ-03-204 triTFA does not induce IKZF1/3 degradation and has anti-cancer activity[1].

Produkteigenschaften

• Molekulargewicht: 1174.97
• Reinheit: 99.87
• Formel: C49H51F9N10O14
• Target-Kategorie: CDK,PROTACs

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound1