BSJ-03-204 (triTFA)

Product Overview

• Article Name: BSJ-03-204 (triTFA)
• Biozol Catalog Number: MCE-HY-136250A
• Supplier Catalog Number: HY-136250A
• Alternative Catalog Number: MCE-HY-136250A-10MG,MCE-HY-136250A-25MG,MCE-HY-136250A-5MG,MCE-HY-136250A-100MG,MCE-HY-136250A-50MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien

Product Description

BSJ-03-204 triTFA is a PROTAC connected by ligands for Cereblon and CDK. BSJ-03-204 triTFA is a potent and selective Palbociclib-based CDK4/6 dual degrader (PROTAC), with IC50s of 26.9 nM and 10.4 nM for CDK4/D1 and CDK6/D1, respectively. BSJ-03-204 triTFA does not induce IKZF1/3 degradation and has anti-cancer activity[1].

Product Properties

• Molecular Weight: 1174.97
• Purity: 99.87
• Formula: C49H51F9N10O14
• Target: CDK,PROTACs

Application Notes

• Application Notes: MCE Product type: Reference compound1