GSK778, CAS [[2451862-42-1]]

Produktübersicht

• Artikelname: GSK778, CAS [[2451862-42-1]]
• Artikelnummer: MCE-HY-136570
• Hersteller Artikelnummer: HY-136570
• Alternativnummer: MCE-HY-136570-5MG,MCE-HY-136570-25MG,MCE-HY-136570-10MMX1ML,MCE-HY-136570-100MG,MCE-HY-136570-10MG,MCE-HY-136570-1MG,MCE-HY-136570-50MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: iBET-BD1

Produktbeschreibung

GSK778 (iBET-BD1), a chemical probe, is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM (BRD2 BD1), 41 nM (BRD3 BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively. GSK778 phenocopies the effects of pan-BET inhibitors in cancer models[1].

Produkteigenschaften

• Molekulargewicht: 511.61
• Reinheit: 99.14
• CAS Nummer: [2451862-42-1]
• Formel: C30H33N5O3
• Target-Kategorie: Apoptosis,Epigenetic Reader Domain

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound