GSK778, CAS [[2451862-42-1]]

Product Overview

• Article Name: GSK778, CAS [[2451862-42-1]]
• Biozol Catalog Number: MCE-HY-136570
• Supplier Catalog Number: HY-136570
• Alternative Catalog Number: MCE-HY-136570-5MG,MCE-HY-136570-25MG,MCE-HY-136570-10MMX1ML,MCE-HY-136570-100MG,MCE-HY-136570-10MG,MCE-HY-136570-1MG,MCE-HY-136570-50MG
• Manufacturer: MedchemExpress
• Category: Biochemikalien
• Alternative Names: iBET-BD1

Product Description

GSK778 (iBET-BD1), a chemical probe, is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM (BRD2 BD1), 41 nM (BRD3 BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively. GSK778 phenocopies the effects of pan-BET inhibitors in cancer models[1].

Product Properties

• Molecular Weight: 511.61
• Purity: 99.14
• CAS Number: [2451862-42-1]
• Formula: C30H33N5O3
• Target: Apoptosis,Epigenetic Reader Domain

Application Notes

• Application Notes: MCE Product type: Reference compound