RP101075, CAS [[1306760-73-5]]

Artikelnummer: MCE-HY-136576
Artikelname: RP101075, CAS [[1306760-73-5]]
Artikelnummer: MCE-HY-136576
Hersteller Artikelnummer: HY-136576
Alternativnummer: MCE-HY-136576-10MG,MCE-HY-136576-50MG,MCE-HY-136576-5MG,MCE-HY-136576-100MG,MCE-HY-136576-25MG,MCE-HY-136576-10MMX1ML
Hersteller: MedchemExpress
Kategorie: Biochemikalien
RP101075, an active metabolite of Ozanimod, is a potent, orally active S1PR (sphingosine-1-phosphate receptor 1) agonist, with an EC50 of 0.27 nM. RP101075 displays >100-fold selectivity over S1PR5 (EC50=5.9 nM) and >10000-fold over S1PR 2, 3, and 4. RP101075 displays superior cardiovascular safety profile[1].
Molekulargewicht: 360.41
Reinheit: 99.19
CAS Nummer: [1306760-73-5]
Formel: C21H20N4O2
Target-Kategorie: Drug Metabolite,LPL Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound