RP101075, an active metabolite of Ozanimod, is a potent, orally active S1PR (sphingosine-1-phosphate receptor 1) agonist, with an EC50 of 0.27 nM. RP101075 displays >100-fold selectivity over S1PR5 (EC50=5.9 nM) and >10000-fold over S1PR 2, 3, and 4. RP101075 displays superior cardiovascular safety profile[1].
Molecular Weight:
360.41
Purity:
99.19
CAS Number:
[1306760-73-5]
Formula:
C21H20N4O2
Target:
Drug Metabolite,LPL Receptor
Application Notes:
MCE Product type: Reference compound
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