RK-582, CAS [[2171388-28-4]]

Produktübersicht

• Artikelname: RK-582, CAS [[2171388-28-4]]
• Artikelnummer: MCE-HY-137849
• Hersteller Artikelnummer: HY-137849
• Alternativnummer: MCE-HY-137849-5MG,MCE-HY-137849-10MG,MCE-HY-137849-100MG,MCE-HY-137849-50MG,MCE-HY-137849-25MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

RK-582 is an orally active, spiroindoline-based selective inhibitor of tankyrase. The IC50s of RK-582 against TNKS1/PARP5A and PARP1 are 36.1 nM and 18.168 nM, respectively. RK-582 inhibits rectal cancer COLO-320DM cells (GI50=0.23 µM) and significantly inhibits tumor growth in a COLO-320DM mouse xenograft model[1].

Produkteigenschaften

• Molekulargewicht: 510.60
• Reinheit: 98.05
• CAS Nummer: [2171388-28-4]
• Formel: C27H35FN6O3
• Target-Kategorie: PARP

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound