EZH2-IN-14, CAS [[1979157-17-9]]

Artikelnummer: MCE-HY-148458
Artikelname: EZH2-IN-14, CAS [[1979157-17-9]]
Artikelnummer: MCE-HY-148458
Hersteller Artikelnummer: HY-148458
Alternativnummer: MCE-HY-148458-5MG,MCE-HY-148458-50MG,MCE-HY-148458-10MG,MCE-HY-148458-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
EZH2-IN-14 is a selective EZH2 (Histone Methyltransferase) inhibitor with an IC50 of 12 nM. EZH2-IN-14 inhibits the methyltransferase activity of EZH2/PRC2 (that is, reducing H3K27me3). EZH2-IN-14 shows >200-fold selective for EZH2 over the highly homologous H3K27 methyltransferase EZH1[1].
Molekulargewicht: 541.69
Reinheit: 99.62
CAS Nummer: [1979157-17-9]
Formel: C31H39N7O2
Target-Kategorie: Histone Methyltransferase
Anwendungsbeschreibung: MCE Product type: Reference compound