HQ005, CAS [[2750644-31-4]]

Artikelnummer: MCE-HY-148523
Artikelname: HQ005, CAS [[2750644-31-4]]
Artikelnummer: MCE-HY-148523
Hersteller Artikelnummer: HY-148523
Alternativnummer: MCE-HY-148523-5MG,MCE-HY-148523-100MG,MCE-HY-148523-10MG,MCE-HY-148523-50MG,MCE-HY-148523-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
HQ005 is a selective CDK12-targeting molecular glue degrader with a DC50 of 41 nM. HQ005 binds to the ATP pocket of CDK12 to mediate CDK12-DDB1 interaction, promote cyclin K ubiquitination, and drive cyclin K proteasomal degradation. HQ005 can be used for the research of cancer, such as non-small cell lung cancer[1][2].
Molekulargewicht: 361.44
Reinheit: 98.56
CAS Nummer: [2750644-31-4]
Formel: C15H15N5O2S2
Target-Kategorie: CDK,Molecular Glues
Anwendungsbeschreibung: MCE Product type: Reference compound