Relutrigine, CAS [[2392951-29-8]]

Produktübersicht

• Artikelname: Relutrigine, CAS [[2392951-29-8]]
• Artikelnummer: MCE-HY-148792
• Hersteller Artikelnummer: HY-148792
• Alternativnummer: MCE-HY-148792-1MG,MCE-HY-148792-5MG,MCE-HY-148792-50MG,MCE-HY-148792-10MG,MCE-HY-148792-10MMX1ML,MCE-HY-148792-25MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien
• Alternative Synonym: PRAX-562

Produktbeschreibung

Relutrigine (PRAX-562) is an orally active inhibitor of persistent sodium channel. Relutrigine potently and preferentially inhibits persistent INa induced by ATX-II (Nav 1.5 activator) or the SCN8A mutation N1768D with IC50 values of 141 nM and 75 nM, respectively. Relutrigine exhibits potent use-dependent block and reduces neuronal intrinsic excitability. Relutrigine has effective anticonvulsant activity[1].

Produkteigenschaften

• Molekulargewicht: 407.27
• Reinheit: 99.13
• CAS Nummer: [2392951-29-8]
• Formel: C15H11F6N5O2
• Target-Kategorie: Sodium Channel

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound