GNE-064, CAS [[1997321-20-6]]

Produktübersicht

• Artikelname: GNE-064, CAS [[1997321-20-6]]
• Artikelnummer: MCE-HY-149026
• Hersteller Artikelnummer: HY-149026
• Alternativnummer: MCE-HY-149026-25MG,MCE-HY-149026-50MG,MCE-HY-149026-10MG,MCE-HY-149026-10MMX1ML,MCE-HY-149026-5MG,MCE-HY-149026-100MG
• Hersteller: MedchemExpress
• Kategorie: Biochemikalien

Produktbeschreibung

GNE-064 (compound 5) is a selective, orally active and highly soluble inhibitor of SMARCA4, SMARCA2 and PBRM1 bromodomains 5. GNE-064 inhibits SMARCA4 with an IC50 of 0.035 µM and inhibits SMARCA2 with an EC50 of 0.10 µM. GNE-064 possess Kds with 0.01, 0.016, 0.018 and 0.049 µM for SMARCA4, SMARCA2, PBRM1 bromodomains 5 and PBRM1 bromodomains 2, repectively. GNE-064 can be used as a chemical probe for the research of agent synthesis[1].

Produkteigenschaften

• Molekulargewicht: 327.38
• Reinheit: 99.65
• CAS Nummer: [1997321-20-6]
• Formel: C17H21N5O2
• Target-Kategorie: Epigenetic Reader Domain

Anwendungsbeschreibung

• Anwendungsbeschreibung: MCE Product type: Reference compound