PROTAC ERalpha Degrader-4, CAS [[2521299-80-7]] Preis auf Anfrage

Artikelnummer: MCE-HY-149295
Artikelname: PROTAC ERalpha Degrader-4, CAS [[2521299-80-7]] Preis auf Anfrage
Artikelnummer: MCE-HY-149295
Hersteller Artikelnummer: HY-149295
Alternativnummer: MCE-HY-149295-5MG,MCE-HY-149295-10MG,MCE-HY-149295-1MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC ERalpha Degrader-4 (Compound ZD12) is a highly potent and selectivePROTAC ERalpha degrader (Ki: 5.08 µM). PROTAC ERalpha Degrader-4 contains OBHSAs, linker and E3 ligase ligands. PROTAC ERalpha Degrader-4 shows excellent cell inhibitory and ERalpha degradation activity against Tamoxifen-sensitive and -resistant ER+ breast cancer (BC) cells and ERalpha-mutated BC cells. PROTAC ERalpha Degrader-4 can induce apoptosis and can be used for cancer research.
Molekulargewicht: 1074.23
Reinheit: 99.06
CAS Nummer: [2521299-80-7]
Formel: C55H62F3N5O10S2
Target-Kategorie: Apoptosis,Estrogen Receptor/ERR,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound