ARD-2051, CAS [[2632305-17-8]]

Artikelnummer: MCE-HY-149862
Artikelname: ARD-2051, CAS [[2632305-17-8]]
Artikelnummer: MCE-HY-149862
Hersteller Artikelnummer: HY-149862
Alternativnummer: MCE-HY-149862-50MG,MCE-HY-149862-1MG,MCE-HY-149862-5MG,MCE-HY-149862-10MG,MCE-HY-149862-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
ARD-2051 is a selective and orally active androgen receptor (AR) proteolysis-targeting chimera degrader. ARD-2051 achieves DC50 values of 0.6 nM for AR protein degradation in both the LNCaP and VCaP prostate cancer cell lines. ARD-2051 exhibits effective anti-tumor activity in VCaP xenograft mice model. ARD-2051 can be used for the research of prostate cancer (Pink: AR ligand (HY-400666), Blue: CRBN Ligand (HY-14658), Black: Linker)[1].
Molekulargewicht: 789.32
Reinheit: 98.57
CAS Nummer: [2632305-17-8]
Formel: C43H45ClN8O5
Target-Kategorie: Androgen Receptor,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound