BI-1622, CAS [[2681392-19-6]]

Artikelnummer: MCE-HY-150023
Artikelname: BI-1622, CAS [[2681392-19-6]]
Artikelnummer: MCE-HY-150023
Hersteller Artikelnummer: HY-150023
Alternativnummer: MCE-HY-150023-5MG,MCE-HY-150023-25MG,MCE-HY-150023-10MMX1ML,MCE-HY-150023-50MG,MCE-HY-150023-100MG,MCE-HY-150023-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
BI-1622 is an orally active, potent and highly selective HER2 (ERBB2) inhibitor, with an IC50 of 7 nM. BI-1622 shows greater than 25-fold selectivity over EGFR. BI-1622 shows high antitumor efficacy in vivo in xenograft mouse tumor models with engineered H2170 and PC9 cells and had a favorable agent metabolism and pharmacokinetics profile[1].
Molekulargewicht: 508.53
Reinheit: 98.97
CAS Nummer: [2681392-19-6]
Formel: C26H24N10O2
Target-Kategorie: Btk,CDK,EGFR,Itk,JAK,PI4K,Raf
Anwendungsbeschreibung: MCE Product type: Reference compound