Nampt degrader-2, CAS [[3035008-40-0]]

Artikelnummer: MCE-HY-152154
Artikelname: Nampt degrader-2, CAS [[3035008-40-0]]
Artikelnummer: MCE-HY-152154
Hersteller Artikelnummer: HY-152154
Alternativnummer: MCE-HY-152154-25MG,MCE-HY-152154-50MG,MCE-HY-152154-5MG,MCE-HY-152154-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Nampt degrader-2 is a fluorescent PROTAC, which efficiently degrades NAMPT with an IC50 of 41.9 nM. Nampt degrader-2 binds to NAMPT and VHL to form a ternary complex and subsequently induced NAMPT degradation via ubiquitin-proteasome system (UPS). Nampt degrader-2 leads to significant reduction of NAD+ and exerts potent antitumor activities[1].
Molekulargewicht: 1052.33
Reinheit: 99.41
CAS Nummer: [3035008-40-0]
Formel: C59H73N9O7S
Target-Kategorie: NAMPT,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound