Zefamenib (BN-104) is an effective selective brain membrane protein inhibitor with oral activity, and its also a Menin inhibitor, it can block the Menin-MLL interaction and leads to the degradation of Menin protein. Zefamenib is a weak hERG inhibitor, with an IC50 greater than 100 µM. Zefamenib has anti-tumor activity and can be used in cancer research, such as for acute myeloid leukemia[1].
Molekulargewicht:
570.66
Reinheit:
99.95
CAS Nummer:
[2938995-50-5]
Formel:
C31H35FN8O2
Target-Kategorie:
Epigenetic Reader Domain,Potassium Channel
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten