FR173657, CAS [[167838-64-4]] Preis auf Anfrage

Artikelnummer: MCE-HY-15791
Artikelname: FR173657, CAS [[167838-64-4]] Preis auf Anfrage
Artikelnummer: MCE-HY-15791
Hersteller Artikelnummer: HY-15791
Alternativnummer: MCE-HY-15791-1UNIT
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: FK-3657
FR173657 is an orally active bradykinin B2 receptor antagonist (IC50: 0.56, 1.5, 2.9 nM for pig, rat, human B2 receptor respectively). FR173657 (p.o.) inhibits BK-induced bronchoconstriction in guinea-pigs (ED50: 0.075 mg/kg). FR173657 (p.o.) also inhibits Carrageenin-induced paw oedema in mice (ED50: 6.8 mg/kg). FR173657 can be used for research of inflammatory disease[1].
Molekulargewicht: 592.47
CAS Nummer: [167838-64-4]
Formel: C30H27Cl2N5O4
Target-Kategorie: Bradykinin Receptor
Anwendungsbeschreibung: MCE Product type: Reference compound