PROTAC K-Ras Degrader-4, CAS [[2938169-99-2]]

Artikelnummer: MCE-HY-159788
Artikelname: PROTAC K-Ras Degrader-4, CAS [[2938169-99-2]]
Artikelnummer: MCE-HY-159788
Hersteller Artikelnummer: HY-159788
Alternativnummer: MCE-HY-159788-5MG,MCE-HY-159788-10MG,MCE-HY-159788-50MG,MCE-HY-159788-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC K-Ras Degrader-4 (Compound 4) is a PROTAC degrader for KRAS that degrades KRASG12D in GP5d and degrades KRASG12V in cell SW620 with DC50s of 1 nM and 13 nM. PROTAC K-Ras Degrader-4 inhibits MAPK signaling pathway[1]. (Pink: ligand for target protein pan-KRAS degrader 1 (HY-162960), Black: linker (HY-159790), Blue: ligand for E3 ligase VHL (HY-W998248))
Molekulargewicht: 989.22
Reinheit: 99.01
CAS Nummer: [2938169-99-2]
Formel: C50H60N12O6S2
Target-Kategorie: PROTACs,Ras
Anwendungsbeschreibung: MCE Product type: Reference compound