VNPP433-3beta, CAS [[1630820-51-7]]

Artikelnummer: MCE-HY-160777
Artikelname: VNPP433-3beta, CAS [[1630820-51-7]]
Artikelnummer: MCE-HY-160777
Hersteller Artikelnummer: HY-160777
Alternativnummer: MCE-HY-160777-5MG,MCE-HY-160777-25MG,MCE-HY-160777-10MG,MCE-HY-160777-1MG,MCE-HY-160777-50MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Alternative Synonym: Galeterone 3beta-imidazole
VNPP433-3beta (Galeterone 3beta-imidazole) is an orally active molecular glue degrader, which degrades androgen receptor (AR) and its splice variants (AR-Vs) and MAP kinase-interacting serine/threonine protein kinase Mnk1/2. VNPP433-3beta induces cell apoptosis. VNPP433-3beta inhibits tumor growth in the CWR22Rv1 xenograft mouse model. VNPP433-3beta can be used for the study of castration resistant prostate cancer (CRPC) and pancreatic ductal adenocarcinoma (PDAC)[1].
Molekulargewicht: 438.61
Reinheit: 98.01
CAS Nummer: [1630820-51-7]
Formel: C29H34N4
Target-Kategorie: Androgen Receptor,Apoptosis,MNK,Molecular Glues
Anwendungsbeschreibung: MCE Product type: Reference compound