C3001a is a selective TREK-1 and TREK-2 channel activator with EC50 values of 12.81 µM and 11.31 µM, respectively. C3001a does not affect other two-pore domain K+ (K2P) channels. C3001a binds to the cryptic binding site formed by P1 and TM4 in TREK-1. C3001a can be used for the study of pain and pancreatitis[1].
Molekulargewicht:
380.46
CAS Nummer:
[2415154-29-7]
Formel:
C21H20N2O3S
Target-Kategorie:
Potassium Channel
Anwendungsbeschreibung:
MCE Product type: Reference compound
* Mehrwertsteuer und Versandkosten nicht enthalten. Irrtümer und Preisänderungen vorbehalten
