C3001a is a selective TREK-1 and TREK-2 channel activator with EC50 values of 12.81 µM and 11.31 µM, respectively. C3001a does not affect other two-pore domain K+ (K2P) channels. C3001a binds to the cryptic binding site formed by P1 and TM4 in TREK-1. C3001a can be used for the study of pain and pancreatitis[1].
Molecular Weight:
380.46
CAS Number:
[2415154-29-7]
Formula:
C21H20N2O3S
Target:
Potassium Channel
Application Notes:
MCE Product type: Reference compound
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