PROTAC KRAS G12D degrader 1, CAS [[3033583-54-6]]

Artikelnummer: MCE-HY-161176
Artikelname: PROTAC KRAS G12D degrader 1, CAS [[3033583-54-6]]
Artikelnummer: MCE-HY-161176
Hersteller Artikelnummer: HY-161176
Alternativnummer: MCE-HY-161176-50MG,MCE-HY-161176-5MG,MCE-HY-161176-1MG,MCE-HY-161176-25MG,MCE-HY-161176-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
PROTAC KRAS G12D degrader 1 is a selective PROTAC KRASG12D degrader. PROTAC KRAS G12D degrader 1 inhibits proliferation of KRASG12D-mutant cells and suppresses ERK phosphorylation. PROTAC KRAS G12D degrader 1 inhibits tumor growth in mice bearing AsPC-1 xenografts. PROTAC KRAS G12D degrader 1 can be used for the study of KRASG12D-driven cancers.(Pink: KRAS ligand (HY-175892), Blue: VHL Ligand (HY-112078), Black: Linker, E3 ligase ligand-linker conjugate (HY-175893))[1].
Molekulargewicht: 1103.33
Reinheit: 98.32
CAS Nummer: [3033583-54-6]
Formel: C59H72F2N10O7S
Target-Kategorie: ERK,PROTACs,Ras
Anwendungsbeschreibung: MCE Product type: Reference compound