PROTAC KRAS G12D degrader 1, CAS [[3033583-54-6]]
Artikelnummer:
MCE-HY-161176
| Artikelname: |
PROTAC KRAS G12D degrader 1, CAS [[3033583-54-6]] |
| Artikelnummer: |
MCE-HY-161176 |
| Hersteller Artikelnummer: |
HY-161176 |
| Alternativnummer: |
MCE-HY-161176-50MG,MCE-HY-161176-5MG,MCE-HY-161176-1MG,MCE-HY-161176-25MG,MCE-HY-161176-10MG |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| PROTAC KRAS G12D degrader 1 is a selective PROTAC KRASG12D degrader. PROTAC KRAS G12D degrader 1 inhibits proliferation of KRASG12D-mutant cells and suppresses ERK phosphorylation. PROTAC KRAS G12D degrader 1 inhibits tumor growth in mice bearing AsPC-1 xenografts. PROTAC KRAS G12D degrader 1 can be used for the study of KRASG12D-driven cancers.(Pink: KRAS ligand (HY-175892), Blue: VHL Ligand (HY-112078), Black: Linker, E3 ligase ligand-linker conjugate (HY-175893))[1]. |
| Molekulargewicht: |
1103.33 |
| Reinheit: |
98.32 |
| CAS Nummer: |
[3033583-54-6] |
| Formel: |
C59H72F2N10O7S |
| Target-Kategorie: |
ERK,PROTACs,Ras |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound |