PROTAC KRAS G12D degrader 1, CAS [[3033583-54-6]]

Catalog Number: MCE-HY-161176
Article Name: PROTAC KRAS G12D degrader 1, CAS [[3033583-54-6]]
Biozol Catalog Number: MCE-HY-161176
Supplier Catalog Number: HY-161176
Alternative Catalog Number: MCE-HY-161176-25MG,MCE-HY-161176-50MG,MCE-HY-161176-1MG,MCE-HY-161176-10MG,MCE-HY-161176-5MG
Manufacturer: MedchemExpress
Category: Biochemikalien
PROTAC KRAS G12D degrader 1 is a selective PROTAC KRASG12D degrader. PROTAC KRAS G12D degrader 1 inhibits proliferation of KRASG12D-mutant cells and suppresses ERK phosphorylation. PROTAC KRAS G12D degrader 1 inhibits tumor growth in mice bearing AsPC-1 xenografts. PROTAC KRAS G12D degrader 1 can be used for the study of KRASG12D-driven cancers.(Pink: KRAS ligand (HY-175892), Blue: VHL Ligand (HY-112078), Black: Linker, E3 ligase ligand-linker conjugate (HY-175893))[1].
Molecular Weight: 1103.33
Purity: 98.32
CAS Number: [3033583-54-6]
Formula: C59H72F2N10O7S
Target: ERK,PROTACs,Ras
Application Notes: MCE Product type: Reference compound1