Nrf2 degrader 1, CAS [[3025286-00-1]]

Artikelnummer: MCE-HY-162307
Artikelname: Nrf2 degrader 1, CAS [[3025286-00-1]]
Artikelnummer: MCE-HY-162307
Hersteller Artikelnummer: HY-162307
Alternativnummer: MCE-HY-162307-5MG,MCE-HY-162307-10MG,MCE-HY-162307-100MG,MCE-HY-162307-50MG,MCE-HY-162307-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
Nrf2 degrader 1 (compound 1) is a PROTAC Nrf2 degrader with a DC50 of 0.1-1 µM in huH1 cells. Nrf2 degrader 1 inhibits cancer cells growth for A549 and LK-2 cells with IC50 values of 100 nM and 40 nM, respectively. Nrf2 degrader 1 can be used for the study of liver cancer, non-small cell lung cancer (NSCLC) and squamous cell carcinoma of lung cancer[1].
Molekulargewicht: 826.92
Reinheit: 99.12
CAS Nummer: [3025286-00-1]
Formel: C45H42N6O8S
Target-Kategorie: Keap1-Nrf2,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound