FOSL1 degrader 1
Artikelnummer:
MCE-HY-162723
| Artikelname: |
FOSL1 degrader 1 |
| Artikelnummer: |
MCE-HY-162723 |
| Hersteller Artikelnummer: |
HY-162723 |
| Alternativnummer: |
MCE-HY-162723-25MG,MCE-HY-162723-5MG,MCE-HY-162723-10MG |
| Hersteller: |
MedchemExpress |
| Kategorie: |
Biochemikalien |
| FOSL1 degrader 1 (4) is a T-5224-PROTAC, potently degrade FOSL1 (AP-1) to suppress cancer stemness gene expression in HNSCC. FOSL1 degrader 1 (4) effectively eliminate HNSCC cancer stem cells to inhibit tumor growth through degrading FOSL1. FOSL1 degrader 1 (4) displays around 30- to 100-fold increased potency over T-5224 (Pink: T-5224 (HY-12270), Black: Linker (HY-130200), Blue: Pomalidomide (HY-10984))[1]. |
| Molekulargewicht: |
1124.19 |
| Reinheit: |
99.47 |
| Formel: |
C58H69N5O18 |
| Target-Kategorie: |
AP-1,PROTACs |
| Anwendungsbeschreibung: |
MCE Product type: Reference compound |