FOSL1 degrader 1

Artikelnummer: MCE-HY-162723
Artikelname: FOSL1 degrader 1
Artikelnummer: MCE-HY-162723
Hersteller Artikelnummer: HY-162723
Alternativnummer: MCE-HY-162723-25MG,MCE-HY-162723-5MG,MCE-HY-162723-10MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
FOSL1 degrader 1 (4) is a T-5224-PROTAC, potently degrade FOSL1 (AP-1) to suppress cancer stemness gene expression in HNSCC. FOSL1 degrader 1 (4) effectively eliminate HNSCC cancer stem cells to inhibit tumor growth through degrading FOSL1. FOSL1 degrader 1 (4) displays around 30- to 100-fold increased potency over T-5224 (Pink: T-5224 (HY-12270), Black: Linker (HY-130200), Blue: Pomalidomide (HY-10984))[1].
Molekulargewicht: 1124.19
Reinheit: 99.47
Formel: C58H69N5O18
Target-Kategorie: AP-1,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound