FOSL1 degrader 1
Catalog Number:
MCE-HY-162723
| Article Name: |
FOSL1 degrader 1 |
| Biozol Catalog Number: |
MCE-HY-162723 |
| Supplier Catalog Number: |
HY-162723 |
| Alternative Catalog Number: |
MCE-HY-162723-25MG,MCE-HY-162723-5MG,MCE-HY-162723-10MG |
| Manufacturer: |
MedchemExpress |
| Category: |
Biochemikalien |
| FOSL1 degrader 1 (4) is a T-5224-PROTAC, potently degrade FOSL1 (AP-1) to suppress cancer stemness gene expression in HNSCC. FOSL1 degrader 1 (4) effectively eliminate HNSCC cancer stem cells to inhibit tumor growth through degrading FOSL1. FOSL1 degrader 1 (4) displays around 30- to 100-fold increased potency over T-5224 (Pink: T-5224 (HY-12270), Black: Linker (HY-130200), Blue: Pomalidomide (HY-10984))[1]. |
| Molecular Weight: |
1124.19 |
| Purity: |
99.47 |
| Formula: |
C58H69N5O18 |
| Target: |
AP-1,PROTACs |
| Application Notes: |
MCE Product type: Reference compound |