G9D-4 (TFA)

Artikelnummer: MCE-HY-162749A
Artikelname: G9D-4 (TFA)
Artikelnummer: MCE-HY-162749A
Hersteller Artikelnummer: HY-162749A
Alternativnummer: MCE-HY-162749A-5MG,MCE-HY-162749A-10MG,MCE-HY-162749A-50MG,MCE-HY-162749A-100MG,MCE-HY-162749A-25MG
Hersteller: MedchemExpress
Kategorie: Biochemikalien
G9D-4 TFA is a G9a PROTAC degrader. G9D-4 TFA induces G9a degradation, reduces H3K9me2 levels, and prevents GLP interference via the CRBN ternary complex, proteasome and ubiquitin-like modification-dependent pathways. G9D-4 TFA exerts antiproliferative activity and induces Apoptosis in pancreatic cancer cells. G9D-4 TFA can be used for research on pancreatic cancer[1].
Molekulargewicht: 1064.24
Reinheit: 99.44
Formel: C55H76F3N9O9
Target-Kategorie: Apoptosis,Histone Methyltransferase,PROTACs
Anwendungsbeschreibung: MCE Product type: Reference compound