G9D-4 (TFA) is a potent PROTAC degrader of G9a, with the DC50 value of 0.1 µM in PANC-1 cells and do not directly perturb GLP protein, with the DC50 of >10 µM. G9D-4 (TFA) plays an important role in pancreatic cancer research (Pink: Ligand for target protein G9a/GLP Inhibitor (HY-15273), Black: Linker, Blue: Ligand for E3 ligase (HY-10984))[1].
Molecular Weight:
1064.24
Purity:
99.44
Formula:
C55H76F3N9O9
Target:
Histone Methyltransferase,PROTACs
Application Notes:
MCE Product type: Reference compound1
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